Why is Understanding Tertiary Structure Important in Drug Design?
In the field of drug design, understanding the tertiary structure of target enzymes is essential. It allows researchers to identify and design inhibitors or activators that can specifically interact with the active site or other crucial regions of the enzyme. By targeting these areas, drugs can modulate the enzyme’s activity, leading to therapeutic effects. Structural insights gained through techniques like X-ray crystallography and NMR spectroscopy are invaluable for rational drug design.
